The use of anabolic steroids has many side effects. Even if athletes follow the correct dosage and adhere to a certain intake pattern, they still have to reckon with small unpleasant consequences. And often when taking steroids, aromatisation occurs, namely the transition from testosterone to oestrogen, and against this background gynaecomastia can develop. To protect against these complications, it is recommended to use aromatase inhibitors after a course of steroids. And among the most effective and efficient is the drug letrozole. It perfectly suppresses all unpleasant effects, restores hormones in the body and normalises testosterone production in athletes.

The prerequisite is taking letrozole during or after a steroid cycle. The drug helps prevent complications and unpleasant consequences. The main thing is to follow the correct dosage regimen and optimal dosage, and it is better to consult a doctor first. You can buy letrozole in the United Kingdom on our website. Only proven and original drugs are offered, which are often used in bodybuilding and other high-performance sports.

Active substance: Letrozole

Letrozole is an aromatase inhibitor that has a strong anti-oestrogenic effect. When taken, it selectively inhibits aromatase (this is an important bioenzyme for the synthesis of oestrogen), this is achieved by highly specific binding to the components of this enzyme. Letrozole inhibits oestrogen biosynthesis in peripheral healthy tissue and tumour tissue.

It helps stop the release of an enzyme in the body, aromatase, which causes the conversion of testosterone to oestradiol. Letrozole preparations are usually used when the course involves the use of medicines with aromatase properties, for example, testosterone esters, methane, etc.

Letrozole is used to control the levels of oestrogen that need to be maintained by their increased production. Proper use of letrozole helps prevent aromatisation and the development of gynaecomastia in athletes, but also increases the growth of free testosterone. If the dosage and the correct administration scheme are observed, drugs with this substance are perfectly tolerated by the body, no unpleasant consequences occur.

ATX code: L02BG04

Structural formula:

Clinical pharmacological group: antitumour hormones and hormone antagonists.

Substances Letrozole

Letrozole -an active ingredient of medicinal products whose use is recommended for the elimination of aromatised effects during the use of anabolic steroids. Based on this, various agents are produced, but they all have the same properties, similar use, indications and contraindications.

Popular manufacturers of drugs containing letrozole include:

Brands Properties
Malaysian Tiger A Malaysian pharmaceutical company that has been supplying medicines for a long time, including for athletes. In their range, there are medicines with Letrozole, they are aromatase inhibitors. They are often used in heavy sports, bodybuilding and weightlifting to reduce the risk of unpleasant consequences after steroid therapy.
Pharmacom Labs A popular pharmaceutical company founded in Moldova in 2006. It manufactures a variety of drugs that are commonly used in sports. Well-known and sought-after cancer drugs include letrozole, which suppresses the aromatising effect after steroid therapy. Reduce the risk of gynaecomastia
Euro Prime Pharmaceuticals A well-known pharmaceutical company founded in Moldova in Chisinau. It is engaged in the development and production of various drugs that are often used in athletes. Aromatase inhibitors with letrozole are popular. They help to cope with all the unpleasant consequences after a steroid cure. Suppress the conversion of testosterone to oestradiol
Magnus Pharmaceuticals A well-known Indian pharmaceutical company that manufactures various types of medicines. Letrozole products are commonly found in pharmacies from this manufacturer and are often used in bodybuilding and other sports. They prevent the development of gynaecomastia. They are used after a steroid cure to suppress side effects and disorders.
Balkan Medicines A popular pharmaceutical company based in Bulgaria. It produces a variety of anabolic steroids used by athletes. Its range also includes medicines containing letrozole, which suppresses the aromatic effect after taking steroids, namely preventing the conversion of testosterone into oestrogen. Reduce the risk of gynaecomastia in bodybuilders and weightlifters.

Release form, packaging and composition of preparations of the active substance letrozole.

In pharmacies, letrozole is often available in tablet form; this is the most popular and sought-after form. Its popularity is due to the fact that the tablets are quite easy to use and no dosage determination is required, as one tablet contains the minimum daily dose.

However, you can also buy letrozole in a solution that comes in ampoules. It has to be injected into a muscle. The dosage is determined individually for each athlete, you should first consult a doctor, they will show you how and where to administer the drug. And it is better to undergo an examination and tests that will help determine exactly what doses of medication with letrozole should be used.

The tablets have a white structure and there are no foreign inclusions on the base. On one side there may be a risk, on the other side there is usually a label from the manufacturer. On the surface there is a shell with an enteric structure, it may have a yellowish hue.

Another form of release is a solution, it has a transparent structure without turbidity and foreign substances. No precipitate forms during storage. The solution may have a yellowish hue and an oily structure. This is because the composition contains a high concentration.

The packaging is made of cardboard and may contain a blister with tablets or a container with ampoules. The name, dosage, description of the medicine and other important information are written on the surface. The package necessarily also contains instructions with a description of the medicinal product.

The composition of the tablets includes the following components:

  • The active substance is letrozole;
  • Auxiliary elements – lactose monohydrate, microcrystalline cellulose, crospovidone, magnesium stearate and others.

The composition of the preparations in the form of a solution includes letrozole. Among the auxiliary components, water for injection, an oil base (olive oil) may be distinguished.

Pharmacological action of letrozole

Letrozole -Aromatase inhibitor commonly used in bodybuilding and heavy sports. After entering the body, the active substance inhibits the conversion of testosterone into oestradiol. Letrozole preparations are used to combat aromatisation by inhibiting the secretion of the aromatase enzyme.

When taking medicines containing letrozole, the release of an enzyme in the body, namely aromatase, is stopped, which leads to the conversion of testosterone into oestradiol. Thanks to its use, it is possible to control the level of oestradiol in the blood, the substance normalises it and prevents a sharp increase.

Letrozole preparations are often prescribed to women for the treatment of breast cancer. They help to suppress the development of the tumour and reduce the risk of gynaecomastia. This is achieved by reducing circulating levels of oestradiol. In the postmenopausal phase, letrozole in a daily dose leads to an 80 % reduction in oestradiol.

Letrozole has no progestogenic, androgenic or oestrogenic activity. When used in therapeutic doses, there is no effect on the secretion of cortisol and aldosterone.

After administration, the active substance letrozole is rapidly absorbed from the gastrointestinal tract. The maximum concentration in the blood is reached within 2 hours after taking the drug. It is recommended to take it on an empty stomach, as food intake may slow down the absorption of the active substance.

What are the benefits of letrozole?

Letrozole drugs are commonly used in bodybuilding when athletes use anabolic steroids. Their use helps to reduce the likelihood of various unpleasant effects. And usually the main purpose is to prevent taste effects when testosterone is converted to oestrogen.

Athletes who take anabolic steroids often struggle with gynaecomastia. This injury is associated with increased growth of the mammary glands. And this is observed due to the fact that testosterone begins to convert into oestrogen. Against this background, serious hormonal disorders can occur, the athlete not only changes his appearance, but also health problems occur, namely constantly rising blood pressure, severe tachycardia, mood swings, potency deterioration, problems in the genital area.

Injectable and tablet letrozole not only helps to eliminate all side effects after a steroid cure, but also has the following positive effects:

  • Stimulates the elimination of stagnant fluid in the body;
  • Suppresses the production of excess female hormones;
  • Stimulates the production of natural testosterone;
  • Reduces the risk of testicular atrophy;
  • Increases libido in men;
  • Protects against the appearance of gynaecomastia;
  • Improves the tone of muscle tissue;
  • Increases the level of anabolic hormones in the blood;
  • Helps reduce the risk of hypertension.

Side effects of letrozole

Side effects should be considered before starting letrozole-containing medicines. They are given in the instructions for use, which are usually included with the medicine in the pack. If you follow all the recommendations and do not exceed the dose, the unpleasant effects will not occur. They can only occur if the regime is violated in case of an overdose.

What side effects may occur when taking medication with letrozole:

  • Headache, dizziness;
  • Frequent mood swings, aggressiveness;
  • Depressed state;
  • Pain in the joints and muscles;
  •  Deterioration in athletic form;
  • Decreased stimulation of metabolic processes;
  • Deterioration of bones, they may lose strength;
  • Decreased libido, deterioration of the reproductive system;
  • Increased blood cholesterol levels;
  • Baldness, deterioration of hair quality;
  • The appearance of rashes on the surface of the skin may be accompanied by itching and redness.
  • Weight gain, but this may be accompanied by a persistent loss of appetite;
  • Anaemia, thrombophlebitis;
  • Injury to the liver.

Letrozole course

You should first learn how to take letrozole. You can find the instructions in the note that comes in the pack of the medicine. It describes the dosage regimen depending on the indication. However, it is better to consult a doctor. He will conduct an examination and select the best application option and dosage.

The use of medication with letrozole is required when taking steroid medication with testosterone. Letrozole can be taken before a course of steroids. However, if there is an increase in the level of aromatisation, this can be detected by testing.

You can take letrozole tablets in the last few weeks of steroid therapy or immediately after stopping steroid use. Bodybuilders should use up to 1-3 mg per day, which can be taken at any time. Even taking a daily dose of 100 micrograms can significantly slow down the effect of the aromatase enzyme’s influence. Do not exceed the recommended dosages, otherwise the risk of unpleasant symptoms and health problems can increase dramatically.

The daily dose should be determined individually for each athlete. But the main thing is not to exceed the recommended dosages of 1-3 mg per day. This dose is sufficient to reduce the development of negative consequences after steroid therapy. The treatment with letrozole can last 1-1.5 months, but you should focus on the general condition. Sometimes the duration of taking medication with letrozole can be prolonged, but in this case it is better to take it every other day.

Indications and contraindications for the use of letrozole

The main indications for the use of medicines containing letrozole are given in the instructions for use. Standard indications include:

  • For the treatment of breast cancer in postmenopausal women;
  • Helps prevent early stages of hormone-positive breast cancer in post-menopausal women after 2-3 years of tamoxifen use;
  • For the treatment of advanced breast cancer in postmenopausal women.

Letrozole is commonly found in bodybuilders and weightlifters. Athletes use drugs containing this substance to reduce the development of gynaecomastia while taking anabolic steroids. The active substance prevents the conversion of testosterone into oestradiol. When using agents containing letrozole, the shock-absorbing effect of anabolic steroids is prevented.

Before taking it, it is important to study the main contraindications of medication with letrozole:

  • Allergic reactions to the main component;
  • The period of pregnancy, breastfeeding;
  •  Liver dysfunction, chronic pathologies;
  • Kidney problems, chronic pathologies;
  • Childhood.

Storage conditions for preparations with the active ingredient letrozole

In order for medicines containing letrozole to retain their basic properties, their therapeutic effects must be stored correctly. It is recommended to store letrozole tablets in a dark place at room temperature, as they do not lose their properties at a temperature of +17 … +25 degrees they do not lose their properties. It is better to store it in a blister pack. The average shelf life is 2 years from the date of issue.

It is recommended to clean preparations in the form of a solution in a cool place, preferably on the bottom shelf of the refrigerator or in the door compartment. The product retains its properties at temperatures from +3 to +7 degrees. Store in an ampoule and in a package. The average life of unopened and unused ampoules is at least two years from the date of issue.

Where to buy Letrozole in Letrozolebuy Anabolic Steroids Shop?

Buy Letrozole in London. You can do this at a pharmacy where medicines of this type are sold. They only offer original products of high quality. But it is better to go to an anabolic steroids pharmacy because they have a wide range of medicines that can be used by athletes. They have all passed the necessary tests, have the relevant certificates and documents confirming high quality and reliability.

If you want to buy Letrozole legally and, above all, not counterfeit, then do not look, but immediately turn to our online shop. We offer original drugs that can eliminate all unpleasant consequences after a course of anabolic steroids. In addition, we offer a wide range of different types of steroids that can be used to build muscle mass, improve appearance, tone the body and increase endurance.

To order Letrozole, you need to fill in the relevant form on the website. It specifies the number of packets and the address to which you want the order delivered. Payment can be made conveniently on the spot. You do not need to present a prescription to make a purchase, but it is better to consult your doctor first so that he or she can select the appropriate application regimen and dosage. Once you have bought Letrozole from our catalogue, delivery is usually fast and takes several days.

On our website you can consult with our managers. They provide the necessary information on all medicines. You can request certificates and documents on medicines from them, all with the appropriate signatures and seals. Our advisors will help you choose the medicine you need and help you buy Letrozole in the United Kingdom.

Letrozole reviews on the active substance

Reviews of letrozole are positive. In sports forums and various services, you can see a lot of comments from athletes who point out that medication with letrozole is really good at preventing unpleasant consequences after taking anabolic steroids. They confirm that taking letrozole reduces the risk of gynaecomastia after anabolic steroids.

Reviews recommend taking medication after consulting specialists. Be sure to follow the doctors’ recommendations and the correct dosage and dosing, otherwise unpleasant effects may occur. Experienced athletes are advised to take the drug immediately after a course of anabolic steroids. It is sufficient to take 1-3 mg per day in the morning or in the evening before going to bed. The average course is 1-1.5 months, depending on the extent of blood depletion.

Reviews of letrozole products can be found on our website. They contain a lot of useful information about the properties of medicines, effects, pharmacological action and schemes for correct use. Athletes believe that medication with letrozole is mandatory, especially when taking a course of anabolic steroids.

Showing 1–16 of 34 results